A Palladium-Catalyzed α-Arylation of Oxindoles with Aryl Tosylates
Publication in refereed journal

香港中文大學研究人員
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其它資訊
摘要A palladium-catalyzed monoselective C3 arylation of 2-oxindoles with aryl tosylates is described. With the Pd/CM-phos catalyst system, the corresponding 3-arylated oxindoles can be obtained in good to excellent yields (≤97%). The reaction conditions are mild (using 0.5 mol % Pd in general and KF as a base), and functional groups such as methyl ester, NH amido, and enolizable keto moieties are found to be compatible.
出版社接受日期25.05.2017
著者DUAN Jindian, KWONG Fuk Yee
期刊名稱Journal of Organic Chemistry
出版年份2017
月份6
日期16
卷號82
期次12
出版社ACS
頁次6468 - 6473
國際標準期刊號0022-3263
語言美式英語

上次更新時間 2021-18-01 於 01:49